# Core Refinement toward Permeable β-Secretase (BACE-1) Inhibitors with Low hERG Activity

**Type:** Papers  
**Canonical URL:** https://scholariq.org/papers/core-refinement-toward-permeable-secretase-bace-1-inhibitors-with-low-herg/

## Facts

| Field | Value |
| --- | --- |
| Author Names | Tobias Ginman,Jenny Viklund,Jonas Malmström,Jan Blid,Rikard Emond,Rickard Forsblom,Anh Johansson,Annika Kers,Fredrik Lake,Fernando W. Sehgelmeble,Karin J. Sterky,Margareta Bergh,Anders Lindgren,Patrik Johansson,Fredrik Jeppsson,Johanna Fälting,Ylva Gravenfors,Fredrik Rahm |
| Citations | 40 |
| DOI | 10.1021/jm3011349 |
| Fields | Biochemistry, Genetics and Molecular Biology,Computer Science,Medicine |
| Open Access | true |
| OA Status | green |
| OA URL | https://doi.org/10.7270/q2ms3wp0 |
| OpenAlex ID | https://openalex.org/W2174168771 |
| PMID | 23126626 |
| Type | article |
| Year | 2012 |

## Paper authors

- [Margareta Bergh](https://scholariq.org/researchers/margareta-bergh/)

## Paper primary topic

- [Computational Drug Discovery Methods](https://scholariq.org/topics/computational-drug-discovery-methods/)

## Paper topics

- [Computational Drug Discovery Methods](https://scholariq.org/topics/computational-drug-discovery-methods/)
- [Chemical Synthesis and Analysis](https://scholariq.org/topics/chemical-synthesis-and-analysis/)
- [Alzheimer's disease research and treatments](https://scholariq.org/topics/alzheimer-s-disease-research-and-treatments/)

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Source: ScholarIQ — public research metadata, principally OpenAlex. See https://scholariq.org/sources/ for provenance and https://scholariq.org/methodology/ for what these figures mean.
