# Discovery of INCB3284, a Potent, Selective, and Orally Bioavailable hCCR2 Antagonist

**Type:** Papers  
**Canonical URL:** https://scholariq.org/papers/discovery-of-incb3284-a-potent-selective-and-orally-bioavailable-hccr2/

## Facts

| Field | Value |
| --- | --- |
| Author Names | Chu‐Biao Xue,Hao Feng,Ganfeng Cao,Taisheng Huang,Joseph Glenn,Rajan Anand,David Meloni,Ke Zhang,Lingquan Kong,Anlai Wang,Yingxin Zhang,Changsheng Zheng,Michael Xia,Lihua Chen,Hiroyuki Tanaka,Qi Han,D. J. Robinson,Dilip Modi,Lou Storace,Lixin Shao,Vaqar Sharief,Mei Li,Laurine G. Galya,Maryanne Covington,Peggy Scherle,Sharon Diamond,Tom Emm,Swamy Yeleswaram,Nancy Contel,Kris Vaddi,Robert Newton,Greg Hollis,Steven Friedman,Brian Metcalf |
| Citations | 48 |
| DOI | 10.1021/ml200030q |
| Fields | Biochemistry, Genetics and Molecular Biology,Medicine |
| Open Access | true |
| OA Status | green |
| OA URL | https://doi.org/10.7270/q2wd4116 |
| OpenAlex ID | https://openalex.org/W2017521644 |
| PMID | 24900329 |
| Type | article |
| Year | 2011 |

## Paper authors

- [Mei Li](https://scholariq.org/researchers/mei-li-2/)

## Paper primary topic

- [Chemokine receptors and signaling](https://scholariq.org/topics/chemokine-receptors-and-signaling/)

## Paper topics

- [Chemokine receptors and signaling](https://scholariq.org/topics/chemokine-receptors-and-signaling/)
- [Monoclonal and Polyclonal Antibodies Research](https://scholariq.org/topics/monoclonal-and-polyclonal-antibodies-research/)
- [Glycosylation and Glycoproteins Research](https://scholariq.org/topics/glycosylation-and-glycoproteins-research/)

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Source: ScholarIQ — public research metadata, principally OpenAlex. See https://scholariq.org/sources/ for provenance and https://scholariq.org/methodology/ for what these figures mean.
