# Inhibitors of Human Immunodeficiency Virus Type 1 (HIV-1) Attachment. 5. An Evolution from Indole to Azaindoles Leading to the Discovery of 1-(4-Benzoylpiperazin-1-yl)-2-(4,7-dimethoxy-1<i>H</i>-pyrrolo\[2,3-<i>c</i>\]pyridin-3-yl)ethane-1,2-dione (BMS-488043), a Drug Candidate That Demonstrates Antiviral Activity in HIV-1-Infected Subjects

**Type:** Papers  
**Canonical URL:** https://scholariq.org/papers/inhibitors-of-human-immunodeficiency-virus-type-1-hiv-1-attachment-5-an/

## Facts

| Field | Value |
| --- | --- |
| Author Names | Tao Wang,Zhiwei Yin,Zhongxing Zhang,John A. Bender,Zhong Yang,Graham Johnson,Zheng Yang,Lisa Zadjura,Celia D’Arienzo,Dawn D. Parker,Christophe Gesenberg,Gregory Yamanaka,Yi-Fei Gong,Hsu‐Tso Ho,Fang Hua,Nannan Zhou,Brian McAuliffe,Betsy J. Eggers,Li Fan,Beata Nowicka-Sans,Ira B. Dicker,Qi Gao,Richard J. Colonno,Pin‐Fang Lin,Nicholas A. Meanwell,John F. Kadow |
| Citations | 99 |
| DOI | 10.1021/jm900843g |
| Fields | Immunology and Microbiology,Medicine |
| Open Access | true |
| OA Status | green |
| OA URL | https://doi.org/10.7270/q2q81d5g |
| OpenAlex ID | https://openalex.org/W1987071206 |
| PMID | 19769332 |
| Type | article |
| Year | 2009 |

## Paper authors

- [Zhongxing Zhang](https://scholariq.org/researchers/zhongxing-zhang/)

## Paper primary topic

- [HIV/AIDS drug development and treatment](https://scholariq.org/topics/hiv-aids-drug-development-and-treatment/)

## Paper topics

- [HIV/AIDS drug development and treatment](https://scholariq.org/topics/hiv-aids-drug-development-and-treatment/)
- [HIV Research and Treatment](https://scholariq.org/topics/hiv-research-and-treatment/)
- [Pneumocystis jirovecii pneumonia detection and treatment](https://scholariq.org/topics/pneumocystis-jirovecii-pneumonia-detection-and-treatment/)

---
Source: ScholarIQ — public research metadata, principally OpenAlex. See https://scholariq.org/sources/ for provenance and https://scholariq.org/methodology/ for what these figures mean.