# SAR Exploration Guided by LE and Fsp <sup>3</sup> : Discovery of a Selective and Orally Efficacious RORγ Inhibitor

**Type:** Papers  
**Canonical URL:** https://scholariq.org/papers/sar-exploration-guided-by-le-and-fsp-sup-3-sup-discovery-of-a-selective-and/

## Facts

| Field | Value |
| --- | --- |
| Author Names | Kazuyuki Hirata,Masayuki Kotoku,Noriyoshi Seki,Takaki Maeba,Katsuya Maeda,Shintaro Hirashima,Takayuki Sakai,Shingo Obika,Akimi Hori,Yasunori Hase,Takayuki Yamaguchi,Yoshiaki Katsuda,Takahiro Hata,Naoki Miyagawa,Kojo Arita,Yukihiro Nomura,Kota Asahina,Yusuke Aratsu,Masafumi Kamada,Tsuyoshi Adachi,Masato Noguchi,Satoki Doi,Paul D. Crowe,Erin K. Bradley,Ruo W. Steensma,Hai‐Yan Tao,Morgan Fenn,Robert E. Babine,Xiaolin Li,Scott M. Thacher,Hiromasa Hashimoto,Makoto Shiozaki |
| Citations | 60 |
| DOI | 10.1021/acsmedchemlett.5b00253 |
| Fields | Biochemistry, Genetics and Molecular Biology,Immunology and Microbiology,Medicine |
| Open Access | true |
| OA Status | green |
| OA URL | https://doi.org/10.7270/q2n58p7p |
| OpenAlex ID | https://openalex.org/W2247001842 |
| PMID | 26819660 |
| Type | article |
| Year | 2015 |

## Paper authors

- [Yukihiro Nomura](https://scholariq.org/researchers/yukihiro-nomura/)

## Paper primary topic

- [Cytokine Signaling Pathways and Interactions](https://scholariq.org/topics/cytokine-signaling-pathways-and-interactions/)

## Paper topics

- [Cytokine Signaling Pathways and Interactions](https://scholariq.org/topics/cytokine-signaling-pathways-and-interactions/)
- [Macrophage Migration Inhibitory Factor](https://scholariq.org/topics/macrophage-migration-inhibitory-factor/)
- [NF-κB Signaling Pathways](https://scholariq.org/topics/nf-b-signaling-pathways/)

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Source: ScholarIQ — public research metadata, principally OpenAlex. See https://scholariq.org/sources/ for provenance and https://scholariq.org/methodology/ for what these figures mean.