# Synthesis and Biological Evaluation

**Type:** Topics  
**Canonical URL:** https://scholariq.org/topics/synthesis-and-biological-evaluation/

## Facts

| Field | Value |
| --- | --- |
| Description | This cluster of papers focuses on the synthesis, biological evaluation, and antimicrobial activity of quinoxaline derivatives. It covers a wide range of topics including the development of new catalysts for synthesis, investigation of their biological activities, and their potential as anticancer agents. |
| Domain | Physical Sciences |
| Field | Chemistry |
| OpenAlex ID | t13160 |
| Works | 61 |

## Topic papers all

Showing 15 of 61.

- [Contribution of Organofluorine Compounds to Pharmaceuticals](https://scholariq.org/papers/contribution-of-organofluorine-compounds-to-pharmaceuticals/)
- [Metabolism and Disposition Kinetics of Nicotine](https://scholariq.org/papers/metabolism-and-disposition-kinetics-of-nicotine/)
- [Pharmacology of Nicotine: Addiction, Smoking-Induced Disease, and Therapeutics](https://scholariq.org/papers/pharmacology-of-nicotine-addiction-smoking-induced-disease-and-therapeutics/)
- [Tobacco-specific nitrosamines, an important group of carcinogens in tobacco and tobacco smoke](https://scholariq.org/papers/tobacco-specific-nitrosamines-an-important-group-of-carcinogens-in-tobacco-and/)
- [Purified protein derivative of Mycobacterium tuberculosis and excretory-secretory antigen(s) of Toxocara canis expand in vitro human T cells with stable and opposite (type 1 T helper or type 2 T helper) profile of cytokine production.](https://scholariq.org/papers/purified-protein-derivative-of-mycobacterium-tuberculosis-and-excretory/)
- [Effect of nicotine and nicotinic receptors on anxiety and depression](https://scholariq.org/papers/effect-of-nicotine-and-nicotinic-receptors-on-anxiety-and-depression/)
- [A Major Role for CYP2A6 in Nicotine C-Oxidation by Human Liver Microsomes](https://scholariq.org/papers/a-major-role-for-cyp2a6-in-nicotine-c-oxidation-by-human-liver-microsomes/)
- [Nicotine metabolism defect reduces smoking](https://scholariq.org/papers/nicotine-metabolism-defect-reduces-smoking/)
- [Free radical formation by antitumor quinones](https://scholariq.org/papers/free-radical-formation-by-antitumor-quinones/)
- [Sulforaphane-induced Cell Death in Human Prostate Cancer Cells Is Initiated by Reactive Oxygen Species](https://scholariq.org/papers/sulforaphane-induced-cell-death-in-human-prostate-cancer-cells-is-initiated-by/)
- [Child and Adolescent Suicide](https://scholariq.org/papers/child-and-adolescent-suicide/)
- [Evidence that mesolimbic dopaminergic activation underlies the locomotor stimulant action of nicotine in rats.](https://scholariq.org/papers/evidence-that-mesolimbic-dopaminergic-activation-underlies-the-locomotor/)
- [NRF2 addiction in cancer cells](https://scholariq.org/papers/nrf2-addiction-in-cancer-cells/)
- [Novel (Rp)-cAMPS Analogs as Tools for Inhibition of cAMP-kinase in Cell Culture](https://scholariq.org/papers/novel-rp-camps-analogs-as-tools-for-inhibition-of-camp-kinase-in-cell-culture/)
- [Benzotriazole: An overview on its versatile biological behavior](https://scholariq.org/papers/benzotriazole-an-overview-on-its-versatile-biological-behavior/)

## Topic primary papers

- [Metabolism and Disposition Kinetics of Nicotine](https://scholariq.org/papers/metabolism-and-disposition-kinetics-of-nicotine/)
- [Tobacco-specific nitrosamines, an important group of carcinogens in tobacco and tobacco smoke](https://scholariq.org/papers/tobacco-specific-nitrosamines-an-important-group-of-carcinogens-in-tobacco-and/)
- [A Major Role for CYP2A6 in Nicotine C-Oxidation by Human Liver Microsomes](https://scholariq.org/papers/a-major-role-for-cyp2a6-in-nicotine-c-oxidation-by-human-liver-microsomes/)
- [Metabolism of nicotine by human liver microsomes: stereoselective formation of trans-nicotine N'-oxide](https://scholariq.org/papers/metabolism-of-nicotine-by-human-liver-microsomes-stereoselective-formation-of/)
- [Digitoxin Inhibits the Growth of Cancer Cell Lines at Concentrations Commonly Found in Cardiac Patients](https://scholariq.org/papers/digitoxin-inhibits-the-growth-of-cancer-cell-lines-at-concentrations-commonly/)
- [Microwave-Assisted Cascade Cycloaddition for C-N Bond Formation: An Approach to the Construction of 1,4,5,6-Tetrahydropyrimidine and 2-Imidazoline Derivatives](https://scholariq.org/papers/microwave-assisted-cascade-cycloaddition-for-c-n-bond-formation-an-approach-to/)
- [(S)-N'-Nitrosonornicotine, a constituent of smokeless tobacco, is a powerful oral cavity carcinogen in rats](https://scholariq.org/papers/s-n-nitrosonornicotine-a-constituent-of-smokeless-tobacco-is-a-powerful-oral/)
- [Characterization and Trypanocidal Activity of Nifurtimox-containing and Empty Nanoparticles of Polyethylc y anoacrylates](https://scholariq.org/papers/characterization-and-trypanocidal-activity-of-nifurtimox-containing-and-empty/)
- [Synthesis and Antiplasmodial Activity of New Indolone <i>N</i>-Oxide Derivatives](https://scholariq.org/papers/synthesis-and-antiplasmodial-activity-of-new-indolone-i-n-i-oxide-derivatives/)
- [Enhancement of antimicrobial activity of pump inhibitors associating drugs](https://scholariq.org/papers/enhancement-of-antimicrobial-activity-of-pump-inhibitors-associating-drugs/)
- [Pharmacokinetics of a nitrofuran compound, nifurtimox, in healthy volunteers.](https://scholariq.org/papers/pharmacokinetics-of-a-nitrofuran-compound-nifurtimox-in-healthy-volunteers/)
- [In vitro and in vivo potentiation by lonidamine of the antitumor effect of adriamycin.](https://scholariq.org/papers/in-vitro-and-in-vivo-potentiation-by-lonidamine-of-the-antitumor-effect-of/)
- [Diversity-Oriented Synthesis of Ketoindoloquinoxalines and Indolotriazoloquinoxalines from 1-(2-Nitroaryl)-2-alkynylindoles](https://scholariq.org/papers/diversity-oriented-synthesis-of-ketoindoloquinoxalines-and/)
- [Diversity Oriented Synthesis of Indoloazepinobenzimidazole and Benzimidazotriazolobenzodiazepine from <i>N</i><sup>1</sup>‐Alkyne‐1,2‐diamines](https://scholariq.org/papers/diversity-oriented-synthesis-of-indoloazepinobenzimidazole-and/)
- [Synthesis and Evaluation of Several New (2-Chloroethyl)nitrosocarbamates as Potential Anticancer Agents](https://scholariq.org/papers/synthesis-and-evaluation-of-several-new-2-chloroethyl-nitrosocarbamates-as/)

---
Source: ScholarIQ — public research metadata, principally OpenAlex. See https://scholariq.org/sources/ for provenance and https://scholariq.org/methodology/ for what these figures mean.
