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ACS Medicinal Chemistry Letters

JournalCitation impact & published research

ACS Medicinal Chemistry Letters is a journal indexed in ScholarIQ from OpenAlex.

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Discovery of Dinaciclib (SCH 727965): A Potent and Selective Inhibitor of Cyclin-Dependent Kinases
Kamil Paruch, Michael P. Dwyer, Carmen Álvarez, Courtney Brown, Tin‐Yau Chan, Ronald J. Doll, Kerry Keertikar, Chad Knutson, Brian A. McKittrick, Jocelyn Rivera, Randall R. Rossman, Gregory A. Tucker, Thierry Fischmann, Alan Hruza, Vincent Madison, Amin A. Nomeir, Yaolin Wang, Paul T. Kirschmeier, Emma Lees, David Parry, Nicole Sgambellone, Wolfgang Seghezzi, Lesley Schultz, Frances Shanahan, Derek Wiswell, Xiaoying Xu, Quiao Zhou, Ray A. James, Vidyadhar M. Paradkar, Haengsoon Park, Laura R. Rokosz, Tara M. Stauffer, Timothy J. Guzi
ACS Medicinal Chemistry Letters. 2010176 Citations
Discovery of Small Molecule RIP1 Kinase Inhibitors for the Treatment of Pathologies Associated with Necroptosis
Philip A. Harris, Deepak Bandyopadhyay, Scott B. Berger, Nino Campobasso, Carol A. Capriotti, Julie A. Cox, Lauren Dare, Joshua N. Finger, Sandra J. Hoffman, Kirsten M. Kahler, Ruth Lehr, John D. Lich, Rakesh Nagilla, Robert T. Nolte, Michael T. Ouellette, Christina Pao, Michelle C. Schaeffer, Angela Smallwood, Helen H. Sun, Barbara A. Swift, Rachel D. Totoritis, Paris Ward, Robert W. Marquis, John Bertin, Peter J. Gough
ACS Medicinal Chemistry Letters. 2013137 CitationsOPEN ACCESS
Crystal Structures of PI3Kα Complexed with PI103 and Its Derivatives: New Directions for Inhibitors Design
Yanlong Zhao, Xi Zhang, Ying‐Yi Chen, Shaoyong Lu, Yuefeng Peng, Xiang Wang, Chengliang Guo, Aiwu Zhou, Jingmiao Zhang, Jingmiao Zhang, Yu Luo, Qiancheng Shen, Jian Ding, Linghua Meng, Jian Zhang, Jian Zhang
ACS Medicinal Chemistry Letters. 2013102 CitationsOPEN ACCESS
Discovery of Brain-Penetrant, Irreversible Kynurenine Aminotransferase II Inhibitors for Schizophrenia
Amy B. Dounay, Marie Anderson, Bruce M. Bechle, Brian Campbell, Michelle M. Claffey, A.G. Evdokimov, Edelweiss Evrard, Kari R. Fonseca, Xinmin Gan, Somraj Ghosh, Matthew M. Hayward, W. Elliott Horner, Jiyoung Kim, Laura A. McAllister, Jayvardhan Pandit, Vanessa Paradis, Vinod D. Parikh, Matthew R. Reese, Suo‐Bao Rong, Michelle A. Salafia, Katherine Schuyten, Christine A. Strick, Jamison B. Tuttle, James J. Valentine, Hong Wang, Laura E. Zawadzke, Patrick R. Verhoest
ACS Medicinal Chemistry Letters. 201291 CitationsOPEN ACCESS
SAR Exploration Guided by LE and Fsp <sup>3</sup> : Discovery of a Selective and Orally Efficacious RORγ Inhibitor
Kazuyuki Hirata, Masayuki Kotoku, Noriyoshi Seki, Takaki Maeba, Katsuya Maeda, Shintaro Hirashima, Takayuki Sakai, Shingo Obika, Akimi Hori, Yasunori Hase, Takayuki Yamaguchi, Yoshiaki Katsuda, Takahiro Hata, Naoki Miyagawa, Kojo Arita, Yukihiro Nomura, Kota Asahina, Yusuke Aratsu, Masafumi Kamada, Tsuyoshi Adachi, Masato Noguchi, Satoki Doi, Paul D. Crowe, Erin K. Bradley, Ruo W. Steensma, Hai‐Yan Tao, Morgan Fenn, Robert E. Babine, Xiaolin Li, Scott M. Thacher, Hiromasa Hashimoto, Makoto Shiozaki
ACS Medicinal Chemistry Letters. 201560 CitationsOPEN ACCESS

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